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团队成员

宾华超

来源: 发布时间:2024-03-11 17:27:38 浏览次数: 【字体:

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宾华超,生物与医药(药物化学)博士,天下足球网中医药创新研究院特聘副研究员。2022年毕业于四川大学。主要研究方向(1)小分子药物的设计、合成与构效关系研究;(2)靶向GPCR的小分子药物以及天然产物的结构优化。以第一/共同第一作者发表论文4篇,以第一发明人申请专利一项。

教育经历

200809-201206:西华大学 制药工程专业;

201209-201506:四川大学华西药学院 药学专业(导师:杨劲松天下足球网);

201809-202112:四川大学生物治疗国家重点实验室 生物与医药专业(导师:杨胜勇天下足球网)。

邮箱:binhuac2024@163.com

科研成果与荣誉

先后在 Nature Communications、European Journal of MedicinalChemistry、Organic Letters 和 Bioorganic & Medicinal Chemistry Letters 期刊上以一作或共同一作发表论文四篇,另有多篇论文以参与作者发表。在校期间,先后取得国家励志奖学金、国家奖学金以及优秀毕业生等荣誉。

(1) Wei Yang, BoMu, Jing You, Chenyu Tian, Huachao Bin, Zhiqiang Xu ,Liting Zhang ,Ronggang Ma, Ming Wu, Guo Zhang, Chong Huang, Linli Li, Zhenhua Shao , Lunzhi Dai ,Laurent Désaubry & Shengyong Yang, Non-classical ferroptosis inhibition by a small moleculetargeting PHB2. Nature Communications, 2022, 13, 7473.(共同一作,2023年影响因子/JCR分区:16.6/Q1)

(2) Huachao Bin, Pei Chen, Ming Wu, Falu Wang, Guifeng Lin, Shulei Pan, Jingming Liu, BoMu, Jinshan Nan, Qiao Huang, Linli Li, Shengyong Yang, Discovery of a potent and highlyselective inhibitor of ataxia telangiectasia mutated and Rad3-Related (ATR) kinase: Structuralactivity relationship and antitumor activity both in vitro and in vivo. European Journal ofMedicinal Chemistry, 2022, 232, 114187.(一作,2023年影响因子/JCR分区:6.7/Q1)

(3) Xing-Yong Liang,?Hua-Chao Bin,?and Jin-Song Yang*. Tuning Effect of Silyl ProtectingGroups on the Glycosylation Reactivity of Arabinofuranosyl Thioglycosides. Organic Letters2013, 15, 2834.(共同一作,2023年影响因子/JCR分区:5.2/Q1)

(4)Pei Chen, Huachao Bin, Yan Jiao, Guifeng Lin, Yun Zhang, Anjie Xia, Zhilin Pan, JingxinQiao, Yinping Guo, Jingming Liu, Yangli Zhou, Linli Li, Discovery of 6,7-dihydro-5H-pyrrolo[3,4-d] pyrimidine derivatives as a new class of ATR inhibitors. Bioorganic & MedicinalChemistry Letters, 2022, 63, 128651.(共同一作,2023年影响因子/JCR分区:2.7/Q2)

(5) Shulei Pan, Liting Zhang, Xinling Luo, Jinshan Nan, Wei Yang, Huachao Bin, Yang Li, QiaoHuang, Tianqi Wang, Zhiling Pan, Bo Mu, Falu Wang, Chenyu Tian, Yang Liu, Linli Li, andShengyong Yang, Structural Optimization and Structure–Activity Relationship Studies of6,6-Dimethyl-4- (phenylamino)-6H-pyrimido[5,4-b][1,4]oxazin-7(8H)-one Derivatives as A NewClass of Potent Inhibitors of Pan-Trk and Their Drug-Resistant Mutants. Journal of MedicinalChemistry, 2022, 65, 2035.(参与作者,2023年影响因子/JCR分区:7.3/Q1)

(6) Yuan Xu, Hua-Chao Bin, Fu Su, Jin-Song Yang*. Stereoselective synthesis of aryl 1,2-cis--furanosides and its application to the synthesis of the carbohydrate portion of antibiotic hygrom-ycin A. Tetrahedron Letters 2017, 58, 1548.(参与作者,2023年影响因子/JCR分区:1.8/Q3)

(7) Qiang-Wei Liu, Hua-Chao Bin, and Jin-Song Yang*. β -Arabinofuranosylation Using5-O-(2-Quinolinecarbonyl) Substituted Ethyl Thioglycoside Donors. Organic Letters 2013, 15,242.(参与作者,2023年影响因子/JCR分区:5.2/Q1)

(8) Xing -Yong Liang, Qiang-Wei Liu, Hua-Chao Bin and Jin-Song Yang*. One-pot synthesisof branched oligosaccharides by use of galacto- and mannopyranosyl thioglycoside diols as keyglyc -osylating agents. Organic & Biomolecular Chemistry 2013, 11, 3903.(参与作者,2023年影响因子/JCR分区:3.2/Q1)



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